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+"WSU-NHL","SIDM00412","909785","UNCLASSIFIED","blood","lymphoid_neoplasm_other","GDSC2","257" +"YAPC","SIDM00411","909904","PAAD","pancreas","pancreas","GDSC1","346" +"YAPC","SIDM00411","909904","PAAD","pancreas","pancreas","GDSC2","282" +"YH-13","SIDM00316","909905","GBM","nervous_system","glioma","GDSC1","352" +"YH-13","SIDM00316","909905","GBM","nervous_system","glioma","GDSC2","282" +"YKG-1","SIDM00315","687592","GBM","nervous_system","glioma","GDSC1","343" +"YKG-1","SIDM00315","687592","GBM","nervous_system","glioma","GDSC2","179" +"YMB-1-E","SIDM01261","1303911","BRCA","breast","breast","GDSC1","135" +"YMB-1-E","SIDM01261","1303911","BRCA","breast","breast","GDSC2","180" +"YT","SIDM00410","946358","ALL","blood","lymphoid_neoplasm_other","GDSC1","387" +"YT","SIDM00410","946358","ALL","blood","lymphoid_neoplasm_other","GDSC2","167" +"ZR-75-30","SIDM00971","909907","BRCA","breast","breast","GDSC1","341" +"ZR-75-30","SIDM00971","909907","BRCA","breast","breast","GDSC2","286" +"huH-1","SIDM00586","1298146","LIHC","digestive_system","liver","GDSC1","352" +"huH-1","SIDM00586","1298146","LIHC","digestive_system","liver","GDSC2","281" +"no-10","SIDM00574","908452","LGG","nervous_system","glioma","GDSC1","393" +"no-10","SIDM00574","908452","LGG","nervous_system","glioma","GDSC2","180" +"no-11","SIDM00573","908450","LGG","nervous_system","glioma","GDSC1","390" +"no-11","SIDM00573","908450","LGG","nervous_system","glioma","GDSC2","179" \ No newline at end of file diff --git a/data/Drug_listTue Dec 3 15_39_27 2024.csv b/data/Drug_listTue Dec 3 15_39_27 2024.csv new file mode 100644 index 0000000..d0d38a6 --- /dev/null +++ b/data/Drug_listTue Dec 3 15_39_27 2024.csv @@ -0,0 +1,701 @@ +Drug Id, Name, Synonyms, Targets, Target pathway, PubCHEM, Datasets, number of cell lines, Screening site +"1242","(5Z)-7-Oxozeaenol","5Z-7-Oxozeaenol, LL-Z1640-2","TAK1","Other, kinases","9863776","GDSC1","899","SANGER" +"1824","123138","","","Unclassified","","GDSC2","717","SANGER" +"1820","123829","","","Unclassified","","GDSC2","717","SANGER" +"1836","150412","","","Unclassified","","GDSC2","717","SANGER" +"179","5-Fluorouracil","5-FU","Antimetabolite (DNA & RNA)","Other","3385","GDSC1","907","MGH" +"1073","5-Fluorouracil","5-FU","Antimetabolite (DNA & RNA)","Other","3385","GDSC2","968","SANGER" +"2156","5-azacytidine","","DNA methyltransferases","Other","","GDSC2","740","SANGER" +"1826","50869","","","Unclassified","","GDSC2","717","SANGER" +"1839","615590","","","Unclassified","","GDSC2","717","SANGER" +"1840","630600","","","Unclassified","","GDSC2","717","SANGER" +"1829","667880","","","Unclassified","","GDSC2","717","SANGER" +"1828","720427","","","Unclassified","","GDSC2","717","SANGER" +"1832","729189","","","Unclassified","","GDSC2","717","SANGER" +"1833","741909","","","Unclassified","","GDSC2","717","SANGER" +"1834","743380","","","Unclassified","","GDSC2","717","SANGER" +"1821","765771","","","Unclassified","","GDSC2","717","SANGER" 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mutant","Metabolism","71299339","GDSC2","893","SANGER" +"2039","AGK2","","BAZ2A, BAZ2B","Chromatin histone acetylation","","GDSC2","933","SANGER" +"1001","AICA Ribonucleotide","AICAR, N1-(b-D-Ribofuranosyl)-5-aminoimidazole-4-carboxamide","AMPK agonist","Metabolism","65110","GDSC1","925","SANGER" +"171","AKT inhibitor VIII","Akti-1/2, KIN001-102","AKT1, AKT2, AKT3","PI3K/MTOR signaling","10196499","GDSC1","877","MGH" +"228","AKT inhibitor VIII","Akti-1/2, KIN001-102","AKT1, AKT2, AKT3","PI3K/MTOR signaling","10196499","GDSC1","913","MGH" +"2045","AMG-319","AMG319","PI3K (beta sparing)","PI3K/MTOR signaling","68947304","GDSC2","950","SANGER" +"272","AR-42","HDAC-42, AR 42, AR42","HDAC1","Chromatin histone acetylation","6918848","GDSC1","899","MGH" +"474","ARRY-520","","KIF11","Mitosis","","GDSC1","899","MGH" +"207","AS601245","","JNK1, JNK2, JNK2","JNK and p38 signaling","10109823","GDSC1","870","MGH" +"224","AS605240","KIN001-173, AS-605240","PI3Kgamma","PI3K/MTOR signaling","5289247","GDSC1","908","MGH" +"381","AST-1306","","EGFR, ERBB4","RTK signaling","","GDSC1","903","MGH" +"219","AT-7519","AT7519","CDK1, CDK2, CDK4, CDK6, CDK9","Cell cycle","11338033","GDSC1","902","MGH" +"2170","AT13148","","AKT1","PI3K/MTOR signaling","","GDSC2","954","SANGER" +"356","AT7867","","AKT","PI3K/MTOR signaling","","GDSC1","919","MGH" +"1184","AZ20","","ATR","Genome integrity","","GDSC1","926","SANGER" +"2109","AZ6102","","TNKS1, TNKS2","WNT signaling","91663328","GDSC2","955","SANGER" +"29","AZ628","AZ-628, AZ 628","BRAF","ERK MAPK signaling","11676786","GDSC1","401","MGH" +"1250","AZ960","AZ 960, AZ-960","JAK2, JAK3","Other, kinases","25099184","GDSC2","892","SANGER" +"1449","AZD1208","SN1028350371","PIM1, PIM2, PIM3","Other, kinases","","GDSC1","921","SANGER" +"1449","AZD1208","SN1028350371","PIM1, PIM2, PIM3","Other, kinases","","GDSC2","716","SANGER" +"1463","AZD1332","SN1061387896","NTRK1, NTRK2, NTRK3","RTK signaling","","GDSC1","919","SANGER" 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+"431","Alisertib","MLN8237","AURKA","Mitosis","","GDSC1","891","MGH" +"1051","Alisertib","MLN8237","AURKA","Mitosis","24771867","GDSC2","949","SANGER" +"1560","Alpelisib","BYL719, BYL-719, NVP-BYL719","PI3Kalpha","PI3K/MTOR signaling","56649450","GDSC2","965","SANGER" +"293","Amuvatinib","MP470, MP 470, MP-470","KIT, PDGFRA, FLT3","RTK signaling","11282283","GDSC1","906","MGH" +"382","Apitolisib","GDC0980","mTOR, PI3K","PI3K/MTOR signaling","","GDSC1","907","MGH" +"427","Ara-G","9-??-D-Arabinofuranosyl guanine","Anti-metabolite","Other","","GDSC1","906","MGH" +"205","Avagacestat","BMS-708163, BMS 708163","Amyloid beta20, Amyloid beta40","Other","46883536","GDSC1","914","MGH" +"1072","Avagacestat","BMS-708163, BMS 708163","Amyloid beta20, Amyloid beta40","Other","46883536","GDSC1","927","SANGER" +"1072","Avagacestat","BMS-708163, BMS 708163","Amyloid beta20, Amyloid beta40","Other","46883536","GDSC2","954","SANGER" +"1021","Axitinib","AG-13736, Inlyta","PDGFR, KIT, VEGFR","RTK signaling","6450551","GDSC1","927","SANGER" +"1021","Axitinib","AG-13736, Inlyta","PDGFR, KIT, VEGFR","RTK signaling","6450551","GDSC2","961","SANGER" +"552","BAM7","","Bax activator","Other","","GDSC1","908","MGH" +"1362","BAY ACCi","","ACACA","Metabolism","","GDSC1","835","SANGER" +"1363","BAY AKT1","","AKT1, AKT2, AKT3","Apoptosis regulation","","GDSC1","835","SANGER" +"178","BAY-61-3606","Syk Inhibitor, BAY-613606","SYK","Other, kinases","10200390","GDSC1","871","MGH" +"1364","BAY-HDAC11_1","","HDAC11","Chromatin histone acetylation","","GDSC1","836","SANGER" +"1365","BAY-HDAC11_2","","HDAC11","Chromatin histone acetylation","","GDSC1","835","SANGER" +"1367","BAY-HDAC11_4","","HDAC11","Chromatin histone acetylation","","GDSC1","835","SANGER" +"1370","BAY-MPS-combo 2 (paclitaxel 1 uM)","","TTK and microtubules","Unclassified","","GDSC1","720","SANGER" +"1369","BAY-MPS-combo-1 (paclitaxel 5 uM)","","TTK and microtubules","Mitosis","","GDSC1","716","SANGER" +"1368","BAY-MPS1","","MPS1","Mitosis","","GDSC1","836","SANGER" +"1585","BDF00022089a","","BRPF1, BRPF2, BRPF3","Chromatin histone acetylation","","GDSC2","717","SANGER" +"1586","BDILV000379a","4-(4-(1-methyl-1H-pyrazol-4-yl)-1-(2-(1-methyl-1H-pyrazol-4-yl)ethyl)-4,5-dihydro-1H-imidazol-5-yl)benzonitrile","BAZ2A, BAZ2B","Chromatin histone acetylation","","GDSC2","717","SANGER" +"1584","BDOCA000347a","4-bromo-N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methylbenzenesulfonamide","BRPF1, BRPF2, BRPF3","Chromatin histone acetylation","","GDSC2","717","SANGER" +"1866","BDP-00009066","","MRCKB_HUMAN","Cytoskeleton","","GDSC2","743","SANGER" +"1847","BEN","","","Unclassified","","GDSC2","717","SANGER" +"60","BI-2536","","PLK1, PLK2, PLK3","Cell cycle","11364421","GDSC1","395","MGH" +"1086","BI-2536","","PLK1, PLK2, PLK3","Cell cycle","11364421","GDSC2","923","SANGER" +"380","BIBF-1120","","VEGFR, PDGFR, FGFR","RTK signaling","","GDSC1","918","MGH" +"2043","BIBR-1532","","TERT","Genome integrity","9927531","GDSC2","952","SANGER" +"279","BIX02189","BIX 02189","MEK5, ERK5","ERK MAPK signaling","46931012","GDSC1","911","MGH" +"203","BMS-345541","BMS345541, IKK Inhibitor 3","IKK1, IKK2","Other, kinases","9813758","GDSC1","916","MGH" +"1249","BMS-345541","","IKK-1, IKK-2","Other","9926054","GDSC2","892","SANGER" +"63","BMS-509744","KIN001-127, ITK inhibitor","ITK","Other, kinases","20635522","GDSC1","398","MGH" +"62","BMS-536924","BMS 536924","IGF1R, IR","IGF1R signaling","10390396","GDSC1","396","MGH" +"1091","BMS-536924","BMS 536924","IGF1R, IR","IGF1R signaling","10390396","GDSC1","909","SANGER" +"1091","BMS-536924","BMS 536924","IGF1R, IR","IGF1R signaling","10390396","GDSC2","958","SANGER" +"184","BMS-754807","BMS754807, BMS 754807","IGF1R, IR","RTK signaling","24785538","GDSC1","865","MGH" +"2171","BMS-754807","BMS-754807","IGF1R, IR","IGF1R signaling","","GDSC2","949","SANGER" +"1998","BPD-00008900","","","Other","","GDSC2","743","SANGER" +"1425","BPTES","SN1041594574","GLS","Other","","GDSC1","916","SANGER" +"222","BX-912","","PDK1 (PDPK1)","Metabolism","11754511","GDSC1","914","MGH" +"1037","BX795","BX-795","TBK1, PDK1 (PDPK1), IKK, AURKB, AURKC","Other, kinases","10077147","GDSC1","932","SANGER" +"1037","BX795","BX-795","TBK1, PDK1 (PDPK1), IKK, AURKB, AURKC","Other, kinases","10077147","GDSC2","225","SANGER" +"274","Belinostat","PXD101, PXD-101","HDAC1","Chromatin histone acetylation","6918638","GDSC1","886","MGH" +"186","Bexarotene","LG-100069, Targretin, Targret, Targrexin, Targretyn, Bexarotenum","Retinioic X receptor (RXR) agonist","Other","82146","GDSC1","861","MGH" +"150","Bicalutamide","ICI-176334, Casodex, Cosudex, ICI 176334","AR","Hormone-related","2375","GDSC1","871","MGH" +"1502","Bicalutamide","ICI-176334, Casodex, Cosudex, ICI 176334","AR","Hormone-related","2375","GDSC1","864","SANGER" +"1502","Bicalutamide","ICI-176334, Casodex, Cosudex, ICI 176334","AR","Hormone-related","2375","GDSC2","225","SANGER" +"190","Bleomycin","","dsDNA break induction","DNA replication","several","GDSC1","856","MGH" +"1812","Bleomycin","","dsDNA break induction","DNA replication","","GDSC2","717","SANGER" +"1392","Bleomycin (10 uM)","","dsDNA break induction","DNA replication","","GDSC1","918","SANGER" +"1378","Bleomycin (50 uM)","","dsDNA break induction","DNA replication","5460769","GDSC1","921","SANGER" +"1378","Bleomycin (50 uM)","","dsDNA break induction","DNA replication","5460769","GDSC2","731","SANGER" +"104","Bortezomib","PS-341, LDP-341, Velcade","Proteasome","Protein stability and degradation","387447","GDSC1","393","MGH" +"1191","Bortezomib","PS-341, LDP-341, Velcade","Proteasome","Protein stability and degradation","387447","GDSC2","957","SANGER" +"1019","Bosutinib","SKI-606, Bosulif","SRC, ABL, TEC","Other, kinases","5328940","GDSC1","932","SANGER" +"1019","Bosutinib","SKI-606, Bosulif","SRC, ABL, TEC","Other, kinases","5328940","GDSC2","949","SANGER" +"376","Brivanib, BMS-540215","","VEGFR, PDGFR","RTK signaling","","GDSC1","918","MGH" +"1581","Bromosporine","ethyl N-[6-(3-methanesulfonamido-4-methylphenyl)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]carbamate","CECR2, BRD2, BRD4, BRD9","Chromatin other","","GDSC2","716","SANGER" +"197","Bryostatin 1","Bryostatin","PKC","Other","5280757","GDSC1","867","MGH" +"1873","Buparlisib","BKM120, NVP-BKM120","PI3Kalpha, PI3Kdelta, PI3Kbeta, PI3Kgamma","PI3K/MTOR signaling","66577015, 16654980","GDSC2","958","SANGER" +"435","C-75","","FAS","Apoptosis regulation","","GDSC1","908","MGH" +"436","CAP-232, TT-232, TLN-232","","Glycolysis","Metabolism","","GDSC1","906","MGH" +"416","CAY10566","","Stearoyl-CoA desaturase","Other","","GDSC1","903","MGH" +"276","CAY10603","","HDAC1, HDAC6","Chromatin histone acetylation","24951314","GDSC1","903","MGH" +"1170","CCT-018159","CCT018159, CCT 018159","HSP90","Protein stability and degradation","5327091","GDSC1","921","SANGER" +"1170","CCT-018159","CCT018159, CCT 018159","HSP90","Protein stability and degradation","5327091","GDSC2","225","SANGER" +"1067","CCT007093","","PPM1D","Cell cycle","2314623","GDSC1","922","SANGER" +"1067","CCT007093","","PPM1D","Cell cycle","2314623","GDSC2","938","SANGER" +"1187","CCT245232","","HSF1","Unclassified","","GDSC1","926","SANGER" +"1188","CCT245467","","HSF1","Unclassified","","GDSC1","925","SANGER" +"449","CD532","","AURKA","Mitosis","","GDSC1","920","MGH" +"1709","CDK9_5038","SN1047483750, CDK9_5038","CDK9","Cell cycle","","GDSC2","716","SANGER" +"1708","CDK9_5576","SN1047226266, CDK9_5576","CDK9","Cell cycle","","GDSC2","716","SANGER" +"54","CGP-082996","CINK4, KIN001-021","CDK4","Cell cycle","24825971","GDSC1","397","MGH" +"53","CGP-60474","KIN001-019, CGP60474, CGP 60474","CDK1,CDK2,CDK5,CDK7,CDK9, PKC","Cell cycle","644215","GDSC1","397","MGH" +"154","CHIR-99021","CT 99021, CHIR99021, CHIR 99021","GSK3A, GSK3B","WNT signaling","9956119","GDSC1","877","MGH" +"1241","CHIR-99021","CT 99021, CHIR99021, CHIR 99021","GSK3A, GSK3B","WNT signaling","9956119","GDSC1","898","SANGER" +"2175","CHIR-99021","CT 99021, CHIR99021, CHIR 99021","GSK3A, GSK3B","WNT signaling","9956119","GDSC2","225","SANGER" +"362","CI-1033","","EGFR, ERBB2, ERBB4","RTK signaling","","GDSC1","916","MGH" +"1015","CI-1040","CI 1040, PD-18435, PD-184352, 212631-79-3","MEK1, MEK2","ERK MAPK signaling","6918454","GDSC1","917","SANGER" +"64","CMK","KIN001-128","RSK2","Other, kinases","16663089","GDSC1","397","MGH" +"152","CP466722","CP-466722, CP 466722, 1080622-86-1","ATM","Genome integrity","44551660","GDSC1","915","MGH" +"255","CP724714","CP-724714","ERBB2","EGFR signaling","9874913","GDSC1","914","MGH" +"415","CPI-613","","Metabo, Mitochondria","Other","","GDSC1","909","MGH" +"2158","CPI-637","","EP300","Chromatin histone methylation","","GDSC2","741","SANGER" +"1071","CRT0105446","","mTOR, LCK","PI3K/MTOR signaling","","GDSC1","923","SANGER" +"1070","CRT0105950","","JNK1, JNK2, JNK3","JNK and p38 signaling","","GDSC1","926","SANGER" +"1183","CRT0160829","","CDC7","DNA replication","","GDSC1","926","SANGER" +"2149","CT7033-2","","KDM4A, KDM4C, KDM4E, KDM3A, KDM6B","Chromatin histone methylation","","GDSC2","741","SANGER" +"273","CUDC-101","CUDC 101","HDAC1-10, EGFR, ERBB2","Other","24756910","GDSC1","893","MGH" +"300","CX-5461","CX5461, CX 5461","RNA Polymerase 1","Other","25257557","GDSC1","906","MGH" +"1615","CZC24832","GTPL6653","PI3Kgamma","PI3K/MTOR signaling","42623951","GDSC2","894","SANGER" +"249","Cabozantinib","BMS-907351, XL-184, Cometriq","VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL","RTK signaling","25102847","GDSC1","911","MGH" +"1003","Camptothecin","Camptothecine, (+)-Camptothecin","TOP1","DNA replication","24360","GDSC2","968","SANGER" +"1136","Capivasertib","AZ5363","AKT","PI3K/MTOR signaling","","GDSC1","924","SANGER" +"1807","Carmustine","","","","","GDSC2","717","SANGER" +"1922","Cediranib","AZD2171, AZD 2171, AZD-2171, Recentin","VEGFR, FLT1, FLT2, FLT3, FLT4, KIT, PDGFRB","RTK signaling","9933475","GDSC2","958","SANGER" +"1114","Cetuximab","Erbitux, IMC-C225, C225, IMC-225, L01XC06","EGFR","EGFR signaling","85668777","GDSC1","862","SANGER" +"1005","Cisplatin","cis-Diammineplatinum(II) dichloride, Platinol, CIS-DDP","DNA crosslinker","DNA replication","84691","GDSC1","934","SANGER" +"1496","Cisplatin","Cisplatin","DNA crosslinker","DNA replication","","GDSC1","919","SANGER" +"1005","Cisplatin","cis-Diammineplatinum(II) dichloride, Platinol, CIS-DDP","DNA crosslinker","DNA replication","84691","GDSC2","760","SANGER" +"37","Crizotinib","Xalkori, PF2341066, PF-2341066, PF 2341066","MET, ALK, ROS1","RTK signaling","11626560","GDSC1","405","MGH" +"1083","Crizotinib","Xalkori, PF2341066, PF-2341066, PF 2341066","MET, ALK, ROS1","RTK signaling","11626560","GDSC2","966","SANGER" +"17","Cyclopamine","","SMO","Other","several","GDSC1","395","MGH" +"1512","Cyclophosphamide","Cytoxan, Neosar, Cyclophosphamid, Procytox, Cyclophosphane","Alkylating agent","DNA replication","2907","GDSC2","957","SANGER" +"1006","Cytarabine","Ara-Cytidine, Arabinosyl Cytosine, U-19920","Antimetabolite","Other","6253","GDSC1","923","SANGER" +"1006","Cytarabine","Ara-Cytidine, Arabinosyl Cytosine, U-19920","Antimetabolite","Other","6253","GDSC2","743","SANGER" +"165","DMOG","Dimethyloxalylglcine","HIF-PH","Metabolism","560326","GDSC1","876","MGH" +"1373","Dabrafenib","GSK2118436, Tafinlar","BRAF","ERK MAPK signaling","44462760","GDSC1","859","SANGER" +"1373","Dabrafenib","GSK2118436, Tafinlar","BRAF","ERK MAPK signaling","44462760","GDSC2","954","SANGER" +"1815","Dacarbazine","DTIC","CP11A","Other","","GDSC2","717","SANGER" +"200","Dacinostat","NVP-LAQ824, LAQ824","HDAC1","Chromatin histone acetylation","6445533","GDSC1","871","MGH" +"1811","Dactinomycin","Actinomycin D","RNA polymerase","Other","","GDSC2","717","SANGER" +"1911","Dactinomycin","Actinomycin D, Cosmegen, Lyovac, Meractinomycin, Ac-De, ActD","RNA polymerase","Other","several","GDSC2","942","SANGER" +"1057","Dactolisib","NVP-BEZ235, BEZ235","PI3K (class 1), MTORC1, MTORC2","PI3K/MTOR signaling","11977753","GDSC1","918","SANGER" +"1057","Dactolisib","NVP-BEZ235, BEZ235","PI3K (class 1), MTORC1, MTORC2","PI3K/MTOR signaling","11977753","GDSC2","958","SANGER" +"1248","Daporinad","APO866, FK866, FK866","NAMPT","Metabolism","6914657","GDSC1","877","SANGER" +"1248","Daporinad","APO866, FK866, FK866","NAMPT","Metabolism","6914657","GDSC2","595","SANGER" +"51","Dasatinib","BMS-354825-03, BMS-354825, Sprycel","ABL, SRC, Ephrins, PDGFR, KIT","RTK signaling","3062316","GDSC1","392","MGH" +"1079","Dasatinib","BMS-354825-03, BMS-354825, Sprycel","ABL, SRC, Ephrins, PDGFR, KIT","Other, kinases","3062316","GDSC2","962","SANGER" +"1827","Dihydrorotenone","","","Unclassified","","GDSC2","715","SANGER" +"1180","Dinaciclib","SCH727965, SCH 727965, SCH-727-965, MK-7965","CDK1, CDK2, CDK5, CDK9","Cell cycle","46926350","GDSC2","891","SANGER" +"1007","Docetaxel","RP-56976, Taxotere","Microtubule stabiliser","Mitosis","148124","GDSC1","933","SANGER" +"1007","Docetaxel","RP-56976, Taxotere","Microtubule stabiliser","Mitosis","148124","GDSC2","967","SANGER" +"1819","Docetaxel","RP-56976, Taxotere","Microtubule stabiliser","Mitosis","","GDSC2","670","SANGER" +"1042","Doramapimod","BIRB-796, BIRB 796","p38, JNK2","JNK and p38 signaling","156422","GDSC1","913","SANGER" +"1042","Doramapimod","BIRB-796, BIRB 796","p38, JNK2","JNK and p38 signaling","156422","GDSC2","955","SANGER" +"133","Doxorubicin","Doxil, Rubex, Adriamycin, Adriablastin, Doxorubicine","Anthracycline","DNA replication","31703","GDSC1","870","MGH" +"1386","Doxorubicin","","Anthracycline","DNA replication","","GDSC1","922","SANGER" +"1407","Dyrk1b_0191","SN1008982787","DYRK1B","Other, kinases","","GDSC1","918","SANGER" +"1069","EHT-1864","EHT 1864","RAC1, RAC2, RAC3","Cytoskeleton","9938202","GDSC1","927","SANGER" +"1069","EHT-1864","EHT 1864","RAC1, RAC2, RAC3","Cytoskeleton","9938202","GDSC2","943","SANGER" +"1237","EPZ004777","EPZ-004777","DOT1L","Chromatin histone methylation","56962336","GDSC2","965","SANGER" +"1563","EPZ5676","EPZ-5676, Pinometostat","DOT1L","Chromatin histone methylation","57345410","GDSC2","962","SANGER" +"1713","ERK_2440","SN1051032892, ERK_2440","ERK1,ERK2","ERK MAPK signaling","","GDSC2","717","SANGER" +"1714","ERK_6604","SN1047587618, ERK_6604","ERK1,ERK2","ERK MAPK signaling","","GDSC2","717","SANGER" +"447","ETP-45835","","MNK1, MNK2","Other, kinases","","GDSC1","919","MGH" +"1712","Eg5_9814","SN1047613775, Eg5_9814","KSP11","Other","","GDSC2","713","SANGER" +"1835","Elephantin","","","Unclassified","","GDSC2","717","SANGER" +"1031","Elesclomol","STA-4783","HSP90","Protein stability and degradation","300471","GDSC1","921","SANGER" +"1031","Elesclomol","STA-4783","HSP90","Protein stability and degradation","300471","GDSC2","225","SANGER" +"172","Embelin","Emberine, Embelic acid","XIAP","Apoptosis regulation","3218","GDSC1","873","MGH" +"88","Entinostat","MS-275","HDAC1, HDAC3","Chromatin histone acetylation","4261","GDSC1","394","MGH" +"1593","Entinostat","MS-275","HDAC1, HDAC3","Chromatin histone acetylation","4261","GDSC2","898","SANGER" +"1630","Entospletinib","GS-9973","SYK","Other, kinases","59473233","GDSC2","894","SANGER" +"229","Enzastaurin","LY317615","PKCB","Other, kinases","176167","GDSC1","912","MGH" +"1413","EphB4_9721","SN1076287848","EPHB4","RTK signaling","","GDSC1","915","SANGER" +"1511","Epirubicin","Ellence, Farmorubicin, IMI-28","Anthracycline","DNA replication","41867","GDSC2","958","SANGER" +"201","Epothilone B","Patupilone, EpoB, EPO906, GNF-PF-193","Microtubule stabiliser","Mitosis","448013","GDSC1","868","MGH" +"1","Erlotinib","Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415","EGFR","EGFR signaling","176870","GDSC1","393","MGH" +"1168","Erlotinib","Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415","EGFR","EGFR signaling","176870","GDSC2","955","SANGER" +"134","Etoposide","Etopophos, Vepesid, Eposin, VP-16","TOP2","DNA replication","36462","GDSC1","879","MGH" +"1419","FEN1_3940","SN1106019609","FEN1","Genome integrity","","GDSC1","912","SANGER" +"1421","FGFR_0939","SN1043317881","FGFR4","RTK signaling","","GDSC1","919","SANGER" +"1422","FGFR_3831","SN1037992934","FGFR1, FGFR2, FGFR3, FGFR4","RTK signaling","","GDSC1","917","SANGER" +"173","FH535","","PPARgamma, PPARdelta","Other","3463933","GDSC1","868","MGH" +"231","FMK","KIN001-242","RSK","Other, kinases","none","GDSC1","784","MGH" +"263","FR-180204","FR 180204, FR180204, ERK Inhibitor II","ERK1, ERK2","ERK MAPK signaling","11493598","GDSC1","912","MGH" +"1128","FS106","","CHEK1","Cell cycle","","GDSC1","925","SANGER" +"1186","FS112","","KS6B1 (p70S6K)","PI3K/MTOR signaling","","GDSC1","925","SANGER" +"166","FTI-277","","Farnesyl-transferase (FNTA)","Other","3005532","GDSC1","880","MGH" +"546","FTY-720","Fingolimod hydrochloride; Gilenya; TDI-132; Imusera; Gilenia","S1P","Other","","GDSC1","909","MGH" +"1198","FY012","","","Unclassified","","GDSC1","914","SANGER" +"1195","FY026","[(para-cymene)osmium(N,N-dimethylphenlyazopyridine)(iodide)]hexafluorophophate","","Unclassified","","GDSC1","915","SANGER" +"1196","FY069","[(biphenyl)osmium(5-fluoro-phenlyazopyridine)(iodide)]hexafluorophophate","","Unclassified","","GDSC1","910","SANGER" +"306","Fedratinib","TG101348, TG-101348, SAR302503, SAR-302503","JAK2","Other, kinases","16722836","GDSC1","914","MGH" +"432","Flavopiridol","","CDK","Cell cycle","","GDSC1","904","MGH" +"1813","Fludarabine","Fludara","Antimetabolite","DNA replication","","GDSC2","717","SANGER" +"308","Foretinib","GSK1363089, XL-880, EXEL-2880, GSK089","MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR","RTK signaling","42642645","GDSC1","909","MGH" +"2040","Foretinib","GSK1363089, XL-880, EXEL-2880, GSK089","MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR","RTK signaling","42642645","GDSC2","953","SANGER" +"1414","Fulvestrant","SN0117217688","ESR1","Hormone-related","","GDSC1","915","SANGER" +"1200","Fulvestrant","Faslodex, ICI-182780","ESR","Hormone-related","104741","GDSC2","963","SANGER" +"1816","Fulvestrant","","ESR","Hormone-related","","GDSC2","717","SANGER" +"1925","GDC0810","GDC-0810, GDC 0810","ESR1, ESR2","Hormone-related","56941241","GDSC2","958","SANGER" +"1926","GNE-317","GNE317, GNE 317","PI3Kalpha","PI3K/MTOR signaling","70676303","GDSC2","944","SANGER" +"52","GNF-2","KIN001-013","BCR-ABL","ABL signaling","5311510","GDSC1","395","MGH" +"1254","GSK-J4","","KDM6B","Chromatin histone methylation","","GDSC1","908","SANGER" +"1583","GSK-LSD1","N-((1R,2S)-2-phenylcyclopropyl)piperidin-4-amine","KDM1","Chromatin histone methylation","","GDSC2","716","SANGER" +"2154","GSK-LSD1-2HCl ","","LSD1","Chromatin histone methylation","","GDSC2","739","SANGER" +"374","GSK1059615","","PI3K","PI3K/MTOR signaling","","GDSC1","904","MGH" +"226","GSK1070916","GSK-1070916","AURKA, AURKC","Mitosis","46885626","GDSC1","868","MGH" +"202","GSK1904529A","GSK-1904529A, GSK 1904529A","IGF1R, IR","RTK signaling","25124816","GDSC1","870","MGH" +"1093","GSK1904529A","GSK-1904529A, GSK 1904529A","IGF1R, IR","IGF1R signaling","25124816","GDSC2","965","SANGER" +"1778","GSK2110183B","","AKT1, AKT2, AKT3","PI3K/MTOR signaling","","GDSC2","717","SANGER" +"1776","GSK2256098C","","FAK1","Cytoskeleton","","GDSC2","717","SANGER" +"1777","GSK2276186C","","JAK1, JAK2, JAK3","Other, kinases","","GDSC2","717","SANGER" +"1927","GSK2578215A","GSK 2578215A, GSK-2578215A","LRRK2","Other, kinases","68107965","GDSC2","958","SANGER" +"1618","GSK2606414","AK175551","PERK","Metabolism","53469448","GDSC2","886","SANGER" +"127","GSK269962A","GSK 269962A","ROCK1, ROCK2","Cytoskeleton","16095342","GDSC1","398","MGH" +"1192","GSK269962A","GSK 269962A","ROCK1, ROCK2","Cytoskeleton","16095342","GDSC1","909","SANGER" +"1192","GSK269962A","GSK 269962A","ROCK1, ROCK2","Cytoskeleton","16095342","GDSC2","268","SANGER" +"1580","GSK2801","1-(7-(2-methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone","","Chromatin other","","GDSC2","717","SANGER" +"2359","GSK2830371","None","WIP1","Other","70983932","GDSC2","731","SANGER" +"1782","GSK2830371A","","PPM1D","Other","","GDSC2","717","SANGER" +"91","GSK319347A","KIN001-135, IKK-3 inhibitor","IKK","Other, kinases","11626927","GDSC1","400","MGH" +"1780","GSK3337463A","","NIK","Other, kinases","","GDSC2","717","SANGER" +"1627","GSK343","GTPL8240, AOB3680, AK175558","EZH2","Chromatin histone methylation","71268957","GDSC2","893","SANGER" +"2037","GSK343","","EZH2","Chromatin histone methylation","","GDSC2","741","SANGER" +"230","GSK429286A","","ROCK1, ROCK2","Cytoskeleton","11373846","GDSC1","913","MGH" +"2110","GSK591","EPZ015866, GSK3203591","PMRT5","Chromatin histone methylation","117072552","GDSC2","954","SANGER" +"1779","GSK626616AC","","DYRK1A","Other, kinases","","GDSC2","717","SANGER" +"177","GSK650394","GSK-650394, GSK 650394","SGK2, SGK3","Other, kinases","25022668","GDSC1","864","MGH" +"326","GSK690693","GSK 690693, GSK-690693","AKT1, AKT2, AKT3","PI3K/MTOR signaling","16725726","GDSC1","910","MGH" +"193","GW-2580","GX2580, CFMS receptor tyrosine kinase inhibitor","CSF1R","RTK signaling","11617559","GDSC1","914","MGH" +"1023","GW441756","GW 441756","NTRK1","RTK signaling","9943465","GDSC1","930","SANGER" +"1023","GW441756","GW 441756","NTRK1","RTK signaling","9943465","GDSC2","953","SANGER" +"87","GW843682X","GW843682X (AN-13)","PLK1","Cell cycle","9826308","GDSC1","394","MGH" +"1830","Gallibiscoquinazole","","","Unclassified","","GDSC2","717","SANGER" +"1010","Gefitinib","ZD-1839, Iressa","EGFR","EGFR signaling","123631","GDSC1","927","SANGER" +"1010","Gefitinib","ZD-1839, Iressa","EGFR","EGFR signaling","123631","GDSC2","958","SANGER" +"135","Gemcitabine","Gemzar, LY-188011","Pyrimidine antimetabolite","DNA replication","60750","GDSC1","859","MGH" +"1393","Gemcitabine","","Pyrimidine antimetabolite","DNA replication","","GDSC1","920","SANGER" +"1190","Gemcitabine","Gemzar, LY-188011","Pyrimidine antimetabolite","DNA replication","60750","GDSC2","960","SANGER" +"225","Genentech Cpd 10","","AURKA, AURKB","Mitosis","none","GDSC1","912","MGH" +"1142","HG-5-113-01","","AURKA","Mitosis","none","GDSC1","491","SANGER" +"1143","HG-5-88-01","","TAK1, M4K2","Other, kinases","none","GDSC1","490","SANGER" +"1204","HG-6-71-01","","DDR1, DDR2, SRC","Other, kinases","","GDSC1","131","SANGER" +"159","HG6-64-1","KIN001-206","BRAF","ERK MAPK signaling","53302361","GDSC1","875","MGH" +"2010","HKMTI-1-005","","","Unclassified","","GDSC2","741","SANGER" +"1232","I-BET-151","GSK12100151A","BRD2, BRD3, BRD4","Chromatin other","","GDSC1","899","SANGER" +"275","I-BET-762","GSK525762A","BRD2, BRD3, BRD4","Chromatin other","46943432","GDSC1","909","MGH" +"1624","I-BET-762","GSK525762A","BRD2, BRD3, BRD4","Chromatin other","46943432","GDSC2","893","SANGER" +"1928","I-BRD9","GSK602, GSK 602, GSK-602","BRD9","Chromatin other","91668541","GDSC2","958","SANGER" +"1531","I-CBP112","","EP300, CBP","Chromatin histone acetylation","","GDSC1","830","SANGER" +"1428","IAP_5620","SN1043546339","IAP","Other","","GDSC1","910","SANGER" +"1428","IAP_5620","SN1043546339","IAP","Other","","GDSC2","714","SANGER" +"1429","IAP_7638","SN1043547481","IAP","Other","","GDSC1","909","SANGER" +"236","IC-87114","","PI3Kdelta","PI3K/MTOR signaling","","GDSC1","913","MGH" +"2011","ICL-SIRT078","","SIR2","Other","","GDSC2","740","SANGER" +"1266","ICL1100013","","N-myristoyltransferase 1/2","Other","","GDSC1","901","SANGER" +"1738","IGF1R_3801","SN1051640224, IGF1R_3801","IGFR1","IGF1R signaling","","GDSC2","716","SANGER" +"1430","IGFR_3801","SN1056768819","IGFR1","IGF1R signaling","","GDSC1","915","SANGER" +"442","IMD-0354","","IKKb","Other, kinases","","GDSC1","912","MGH" +"1230","IOX2","IOX-2, IOX 2, AK176060","EGLN1","Other","54685215","GDSC1","913","SANGER" +"2174","IOX2","IOX-2, IOX 2, AK176060","EGLN1","Other","54685215","GDSC2","225","SANGER" +"176","IPA-3","IPA 3","PAK1","Cytoskeleton","521106","GDSC1","869","MGH" +"1716","IRAK4_4710","SN1050852374, IRAK4_4710","IRAK4","Other, kinases","","GDSC2","717","SANGER" +"1576","IWP-2","Wnt Inhibitor IWP-2","PORCN","WNT signaling","2155128","GDSC2","893","SANGER" +"1799","Ibrutinib","PCI-32765, CRA-032765, PCI-32765-00","BTK","Other, kinases","24821094","GDSC2","890","SANGER" +"238","Idelalisib","CAL-101, Zydelig","PI3Kdelta","PI3K/MTOR signaling","11625818","GDSC1","914","MGH" +"34","Imatinib","Gleevec, STI-571","ABL, KIT, PDGFR","Other, kinases","5291","GDSC1","404","MGH" +"1924","Ipatasertib","GDC0068, GDC 0068, GDC-0068","AKT1, AKT, AKT3","PI3K/MTOR signaling","24788740","GDSC2","958","SANGER" +"1088","Irinotecan","Camptosar, (+)-Irinotecan, Irinotecanum, irinotecan hydrochloride","TOP1","DNA replication","60838","GDSC2","965","SANGER" +"208","Ispinesib Mesylate","SB-715992","KSP","Mitosis","6450816","GDSC1","911","MGH" +"1433","JAK1_3715","SN1042605297","JAK1","Other, kinases","","GDSC1","920","SANGER" +"1718","JAK1_8709","SN1049200060, JAK1_8709","JAK1","Other, kinases","","GDSC2","717","SANGER" +"1434","JAK3_7406","SN1014281280","JAK3","Other, kinases","","GDSC1","918","SANGER" +"1739","JAK_8517","SN1066590414, JAK_8517","JAK1, JAK2","Other, kinases","","GDSC2","717","SANGER" +"284","JNJ38877605","","MET","RTK signaling","","GDSC1","917","MGH" +"1043","JNK Inhibitor VIII","","JNK","JNK and p38 signaling","11624601","GDSC1","929","SANGER" +"1043","JNK Inhibitor VIII","","JNK","JNK and p38 signaling","11624601","GDSC2","950","SANGER" +"157","JNK-9L","KIN001-204, JNK inhibitor 9l","JNK2, JNK3","JNK and p38 signaling","25222038","GDSC1","879","MGH" +"1205","JNK-9L","","BAZ2A, BAZ2B","","","GDSC1","131","SANGER" +"163","JQ1","JQ-1, (+)-JQ-1","BRD2, BRD3, BRD4, BRDT","Chromatin other","46907787","GDSC1","879","MGH" +"1218","JQ1","JQ-1, (+)-JQ-1","BRD2, BRD3, BRD4, BRDT","Chromatin other","46907787","GDSC1","898","SANGER" +"2172","JQ1","JQ-1, (+)-JQ-1","BRD2, BRD3, BRD4, BRDT","Chromatin other","46907787","GDSC2","949","SANGER" +"164","JQ12","","HDAC1, HDAC2","Chromatin histone acetylation","none","GDSC1","873","MGH" +"256","JW-7-24-1","","LCK","Other, kinases","none","GDSC1","914","MGH" +"83","JW-7-52-1","NA","MTOR","PI3K/MTOR signaling","49836027","GDSC1","382","MGH" +"289","KIN001-042","","GSK3B","WNT signaling","","GDSC1","917","MGH" +"286","KIN001-236","","HDAC6, HDAC10","Chromatin histone acetylation","none","GDSC1","912","MGH" +"287","KIN001-244","PDK1 inhibitor 7","PDK1","Other, kinases","56965967","GDSC1","911","MGH" +"290","KIN001-260","Bayer IKKb inhibitor, ACHP","CDC7","DNA replication","10451420","GDSC1","911","MGH" +"291","KIN001-266","","CDC7","DNA replication","44143370","GDSC1","911","MGH" +"345","KIN001-270","CDK9 inhibitor, CDK9-IN-1","CDK9","Other","66577006","GDSC1","912","MGH" +"1855","KRAS (G12C) Inhibitor-12","GTPL8020","KRAS (G12C)","ERK MAPK signaling","73555129","GDSC2","894","SANGER" +"1030","KU-55933","KU55933","ATM","Genome integrity","5278396","GDSC1","931","SANGER" +"1030","KU-55933","KU55933","ATM","Genome integrity","5278396","GDSC2","955","SANGER" +"1185","KU-60019","","ATM","Genome integrity","","GDSC1","925","SANGER" +"563","Kobe2602","","RAS effector","RTK signaling","","GDSC1","907","MGH" +"1831","L-Oxonoreleagnine","","","Unclassified","","GDSC2","717","SANGER" +"439","LCL161","","XIAP, cIAP1, cIAP2","Apoptosis regulation","","GDSC1","905","MGH" +"1557","LCL161","","XIAP, IAP1, IAP2","Apoptosis regulation","24737642","GDSC2","893","SANGER" +"478","LDN-193189","","BMP","Other","","GDSC1","907","MGH" +"192","LFM-A13","DDE-28","BTK","Other, kinases","54676905","GDSC1","871","MGH" +"573","LGK974","","PORCN","WNT signaling","","GDSC1","905","MGH" +"1598","LGK974","LGK-974","PORCN","WNT signaling","46926973","GDSC2","964","SANGER" +"406","LIMK1 inhibitor BMS4","","LIMK1","Cytoskeleton","","GDSC1","919","MGH" +"2107","LJI308","","RSK2, RSK1, RSK3","PI3K/MTOR signaling","118704762","GDSC2","954","SANGER" +"1783","LMB_AB1","","ADRA1A, ADRB1","Other","","GDSC2","717","SANGER" +"1784","LMB_AB2","","GADD34","Unclassified","","GDSC2","717","SANGER" +"1785","LMB_AB3","","PPP1R15B","Other","","GDSC2","717","SANGER" +"1843","LMP744","MJ-III-65","TOP1","DNA replication","","GDSC2","717","SANGER" +"1852","LY2109761","5XE","TGFB1","Other","11655119","GDSC2","892","SANGER" +"119","Lapatinib","Tykerb, Tyverb","EGFR, ERBB2","RTK signaling","208908","GDSC1","395","MGH" +"1558","Lapatinib","Tykerb, Tyverb","EGFR, ERBB2","EGFR signaling","208908","GDSC2","966","SANGER" +"1578","Leflunomide","Sulol, SU-101, HWA-486, Arava","Pyrimidine synthesis inhibitor","DNA replication","3899","GDSC2","894","SANGER" +"1020","Lenalidomide","CDC-501, CC-5013, Revlimid","CRBN","Protein stability and degradation","216326","GDSC1","933","SANGER" +"1020","Lenalidomide","CDC-501, CC-5013, Revlimid","CRBN","Protein stability and degradation","216326","GDSC2","949","SANGER" +"1024","Lestaurtinib","CEP-701, SP-924, SPM-924, A-154475, KT-555","FLT3, JAK2, NTRK1, NTRK2, NTRK3","Other, kinases","126565","GDSC1","929","SANGER" +"1024","Lestaurtinib","CEP-701, SP-924, SPM-924, A-154475, KT-555","FLT3, JAK2, NTRK1, NTRK2, NTRK3","Other, kinases","126565","GDSC2","947","SANGER" +"277","Linifanib","ABT-869, ABT 869","VEGFR1, VEGFR2, VEGFR3, CSF1R, FLT3, KIT","RTK signaling","11485656","GDSC1","914","MGH" +"185","Linsitinib","OSI-906, ASP-7487","IGF1R","IGF1R signaling","11640390","GDSC1","867","MGH" +"1510","Linsitinib","OSI-906, ASP-7487","IGF1R","IGF1R signaling","11640390","GDSC2","966","SANGER" +"194","Luminespib","AUY922, VER-52296,NVP-AUY922, AUY","HSP90","Protein stability and degradation","10096043","GDSC1","862","MGH" +"1559","Luminespib","AUY922, VER-52296,NVP-AUY922, AUY","HSP90","Protein stability and degradation","10096043","GDSC2","964","SANGER" +"1436","MCT1_6447","SN0177231247","MCT1","Cell cycle","","GDSC1","897","SANGER" +"1437","MCT4_1422","SN1043999849","MCT4","Other","","GDSC1","918","SANGER" +"9","MG-132","LLL cpd, MG 132, MG132","Proteasome, CAPN1","Protein stability and degradation","462382","GDSC1","398","MGH" +"1862","MG-132","LLL cpd, MG 132, MG132","Proteasome, CAPN1","Protein stability and degradation","462382","GDSC2","969","SANGER" +"446","MIM1","","MCL-1","Apoptosis regulation","","GDSC1","901","MGH" +"1996","MIM1","MIM 1, MIM-1","MCL1","Apoptosis regulation","16241412","GDSC2","743","SANGER" +"1931","MIRA-1","MIRA 1, MIRA1, NSC19630, NSC-19630, NSC 19630","TP53","p53 pathway","227681","GDSC2","966","SANGER" +"1179","MK-1775","AZD1775, Adavosertib","WEE1, PLK1","Cell cycle","24856436","GDSC2","967","SANGER" +"1053","MK-2206","MK 2206, MK2206","AKT1, AKT2","PI3K/MTOR signaling","46930998","GDSC1","888","SANGER" +"1053","MK-2206","MK 2206, MK2206","AKT1, AKT2","PI3K/MTOR signaling","46930998","GDSC2","968","SANGER" +"2046","MK-8776","SCH900776","CHEK1, CHEK2, CDK2","Cell cycle","16224745","GDSC2","952","SANGER" +"1629","ML323","GTPL7898, AOB2313,","USP1, UAF1","Protein stability and degradation","60167849","GDSC2","891","SANGER" +"1854","MN-64","","TNKS1, TNKS2","WNT signaling","2802462","GDSC2","894","SANGER" +"294","MPS-1-IN-1","","MPS1","Mitosis","25195352","GDSC1","910","MGH" +"292","Masitinib","AB1010, Masivet","KIT, PDGFRA, PDGFRB","RTK signaling","10074640","GDSC1","913","MGH" +"410","MetAP2 Inhibitor, A832234","","MetAP2","Other","","GDSC1","903","MGH" +"1008","Methotrexate","Abitrexate, Amethopterin, Rheumatrex, Trexall, Folex","Antimetabolite","DNA replication","126941","GDSC1","933","SANGER" +"1008","Methotrexate","Abitrexate, Amethopterin, Rheumatrex, Trexall, Folex","Antimetabolite","DNA replication","126941","GDSC2","881","SANGER" +"153","Midostaurin","PKC412, benzoylstaurosporine, CGP-41251","PKC, PPK, FLT1, c-FGR, others","Other","several","GDSC1","881","MGH" +"1048","Mirin","","MRE11","Genome integrity","none","GDSC1","846","SANGER" +"1048","Mirin","","MRE11","Genome integrity","none","GDSC2","894","SANGER" +"136","Mitomycin-C","Mytozytrex, NSC-26980, MMC, Mitosol, Mitozytrex","DNA crosslinker","DNA replication","5746","GDSC1","870","MGH" +"1810","Mitoxantrone","","TOP2","DNA replication","","GDSC2","717","SANGER" +"1029","Motesanib","AMG-706, AMG 706, AMG706","VEGFR, RET, KIT, PDGFR","RTK signaling","11667893","GDSC1","927","SANGER" +"1029","Motesanib","AMG-706, AMG 706, AMG706","VEGFR, RET, KIT, PDGFR","RTK signaling","11667893","GDSC2","949","SANGER" +"2055","Mycophenolic acid","","","Unclassified","","GDSC2","737","SANGER" +"2499","N-acetyl cysteine","NAC","Metabolism","Metabolism","None","GDSC2","735","SANGER" +"1251","N22899-6-C1","","Peptidyl arginine deaminase (PAD)","Unclassified","","GDSC1","913","SANGER" +"1252","N23918-95-7","","JMJ histone demethylase","Chromatin histone methylation","","GDSC1","913","SANGER" +"1253","N24798-49-A1","","JMJ histone demethylase","Chromatin histone methylation","","GDSC1","908","SANGER" +"1999","N25720-51-A1","","","Unclassified","","GDSC2","742","SANGER" +"2000","N27922-53-1","","","Unclassified","","GDSC2","743","SANGER" +"2003","N29087-69-1","","","Unclassified","","GDSC2","743","SANGER" +"2002","N30652-18-1","","","Unclassified","","GDSC2","743","SANGER" +"260","NG-25","NG25","TAK1, M4K2","Other, kinases","53340664","GDSC1","912","MGH" +"1167","NG-25","","TAK1","Unclassified","","GDSC1","96","SANGER" +"257","NPK76-II-72-1","","PLK3","Cell cycle","none","GDSC1","911","MGH" +"269","NSC-207895","XI-006, NSC207895","MDM4","p53 pathway","42640","GDSC1","908","MGH" +"147","NSC-87877","NSC 87877","SHP-1 (PTPN6), SHP-2 (PTPN11)","Other","5459322","GDSC1","877","MGH" +"461","NSC319726","","P53 Mut specific","p53 pathway","","GDSC1","873","MGH" +"1038","NU7441","KU-57788, NU-7432, NU-7741","DNAPK","Genome integrity","11327430","GDSC1","926","SANGER" +"1038","NU7441","KU-57788, NU-7432, NU-7741","DNAPK","Genome integrity","11327430","GDSC2","945","SANGER" +"1932","NVP-ADW742","NVP ADW742, NVPADW742","IGF1R","IGF1R signaling","9825149","GDSC2","958","SANGER" +"295","NVP-BHG712","BHG712","EPHB4, RAF, SRC, ABL","Other, kinases","16747388","GDSC1","912","MGH" +"35","NVP-TAE684","NVP-TAE 684, TAE684, TAE-684","ALK","RTK signaling","16038120","GDSC1","403","MGH" +"1011","Navitoclax","ABT-263, ABT263, ABT 263","BCL2, BCL-XL, BCL-W","Apoptosis regulation","24978538","GDSC1","928","SANGER" +"1011","Navitoclax","ABT-263, ABT263, ABT 263","BCL2, BCL-XL, BCL-W","Apoptosis regulation","24978538","GDSC2","967","SANGER" +"1814","Nelarabine","Atriance, Arranon","","DNA replication","","GDSC2","716","SANGER" +"1013","Nilotinib","Tasigna, AMN 107","ABL","ABL signaling","644241","GDSC1","933","SANGER" +"1013","Nilotinib","Tasigna, AMN 107","ABL","ABL signaling","644241","GDSC2","955","SANGER" +"1177","Niraparib","MK-4827, MK4827","PARP1, PARP2","Genome integrity","24958200","GDSC2","894","SANGER" +"1047","Nutlin-3a (-)","","MDM2","p53 pathway","11433190","GDSC1","933","SANGER" +"1047","Nutlin-3a (-)","","MDM2","p53 pathway","11433190","GDSC2","968","SANGER" +"1853","OF-1","","BRPF1B, BRPF2","Chromatin histone acetylation","35397514","GDSC2","894","SANGER" +"299","OSI-027","A-1065-5","MTORC1, MTORC2","PI3K/MTOR signaling","44224160","GDSC1","900","MGH" +"1594","OSI-027","A-1065-5","MTORC1, MTORC2","PI3K/MTOR signaling","44224160","GDSC2","960","SANGER" +"298","OSI-930","OSI 930 OSI930","KIT, VEGFR2","RTK signaling","9868037","GDSC1","913","MGH" +"167","OSU-03012","AR-12, OSU 03012, OSU03012, PDK1 inhibitor AR-12","PDK1 (PDPK1)","Metabolism","10027278","GDSC1","870","MGH" +"1626","OTX015","Birabresib, OTX-015, MK-8628","BRD2, BRD3, BRD4","Chromatin other","9936746","GDSC2","893","SANGER" +"182","Obatoclax Mesylate","GX15-070MS, Obatoclax, GX15-070","BCL2, BCL-XL, BCL-W, MCL1","Apoptosis regulation","11404337","GDSC1","862","MGH" +"1068","Obatoclax Mesylate","GX15-070MS, Obatoclax, GX15-070","BCL2, BCL-XL, BCL-W, MCL1","Apoptosis regulation","11404337","GDSC2","785","SANGER" +"1017","Olaparib","AZD2281, KU0059436, Lynparza","PARP1, PARP2","Genome integrity","23725625","GDSC1","932","SANGER" +"1495","Olaparib","AZD2281, KU0059436, Lynparza","PARP1, PARP2","Genome integrity","23725625","GDSC1","895","SANGER" +"1017","Olaparib","AZD2281, KU0059436, Lynparza","PARP1, PARP2","Genome integrity","23725625","GDSC2","967","SANGER" +"283","Omipalisib","GSK2126458, GSK-2126458, EX-8678, GSK458","PI3K (class 1), MTORC1, MTORC2","PI3K/MTOR signaling","25167777","GDSC1","914","MGH" +"1919","Osimertinib","AZD9291, AZD 9291, AZD-9291, Tagrisso, Mereletinib","EGFR","EGFR signaling","71496458","GDSC2","957","SANGER" +"1089","Oxaliplatin","Eloxatin","DNA alkylating agent","DNA replication","5310940","GDSC2","967","SANGER" +"1806","Oxaliplatin","","DNA alkylating agent","DNA replication","","GDSC2","717","SANGER" +"1933","P22077","P 22077, P-22077","USP7, USP47","Protein stability and degradation","46931953","GDSC2","958","SANGER" +"175","PAC-1","GTPL5238","Procaspase-3, Procaspase-7","Apoptosis regulation","6753378","GDSC1","857","MGH" +"1730","PAK_5339","SN1046290829, PAK_5339","PAK1, PAK2","Cytoskeleton","","GDSC2","716","SANGER" +"1459","PARP_0108","SN1044053371","PARP1, PARP2, PARP6","Genome integrity","","GDSC1","918","SANGER" +"1460","PARP_9482","SN1031920820","PARP1, PARP2, PARP5a","Genome integrity","","GDSC1","915","SANGER" +"1458","PARP_9495","SN1024601395","PARP1, PARP2, PARP7","Genome integrity","","GDSC1","911","SANGER" +"2145","PBD-288","","","Unclassified","","GDSC2","741","SANGER" +"1621","PCI-34051","AK298746","HDAC8, HDAC6, HDAC1","Chromatin histone acetylation","24753719","GDSC2","894","SANGER" +"1060","PD0325901","PD-0325901, PD 0325901","MEK1, MEK2","ERK MAPK signaling","9826528","GDSC1","918","SANGER" +"1060","PD0325901","PD-0325901, PD 0325901","MEK1, MEK2","ERK MAPK signaling","9826528","GDSC2","968","SANGER" +"1049","PD173074","PD-173074, PD 173074","FGFR1, FGFR2, FGFR3","RTK signaling","1401","GDSC1","932","SANGER" +"1049","PD173074","PD-173074, PD 173074","FGFR1, FGFR2, FGFR3","RTK signaling","1401","GDSC2","967","SANGER" +"363","PF-00299804","","EGFR, ERBB2, ERBB4","RTK signaling","","GDSC1","909","MGH" +"1129","PF-4708671","PF 4708671, PF4708671","S6K1","PI3K/MTOR signaling","51371303","GDSC1","916","SANGER" +"1129","PF-4708671","PF 4708671, PF4708671","S6K1","PI3K/MTOR signaling","51371303","GDSC2","268","SANGER" +"158","PF-562271","PF-00562271","FAK, FAK2","Cytoskeleton","11713159","GDSC1","864","MGH" +"1219","PFI-1","","BRD4","Chromatin other","71271629","GDSC1","914","SANGER" +"2173","PFI-1","","BRD4","Chromatin other","71271629","GDSC2","946","SANGER" +"1530","PFI-3","BDF00016096","PB1, SMARCA4, SMARCA2","Chromatin other","78243717","GDSC1","834","SANGER" +"1620","PFI3","PFI-3, PFI 3, AOB2221","Polybromo 1, SMARCA4, SMARCA2","Chromatin other","78243717","GDSC2","894","SANGER" +"6","PHA-665752","PHA665752, PHA 665752","MET","RTK signaling","10461815","GDSC1","405","MGH" +"301","PHA-793887","PHA793887, PHA 793887","CDK2, CDK7, CDK5","Cell cycle","46191454","GDSC1","912","MGH" +"302","PI-103","PI-103, PI103, PI 103","PI3Kalpha, DAPK3, CLK4, PIM3, HIPK2","Other, kinases","9884685","GDSC1","902","MGH" +"1446","PI3Ka_4409","SN1037097676","PI3Kalpha, PI3Kdelta","PI3K/MTOR signaling","","GDSC1","913","SANGER" +"303","PIK-93","PIK 93, PIK93","PK3CG","PI3K/MTOR signaling","6852167","GDSC1","911","MGH" +"1451","PLK_6522","SN1077317349","PLK1, PLK2, PLK3","Cell cycle","","GDSC1","903","SANGER" +"1036","PLX-4720","PLX4720, PLX 4720","BRAF","ERK MAPK signaling","24180719","GDSC1","930","SANGER" +"1371","PLX-4720","PLX4720, PLX 4720","BRAF","ERK MAPK signaling","24180719","GDSC1","913","SANGER" +"1036","PLX-4720","PLX4720, PLX 4720","BRAF","ERK MAPK signaling","24180719","GDSC2","961","SANGER" +"2148","POMHEX","","","Unclassified","","GDSC2","741","SANGER" +"1131","PRIMA-1MET","Prima 1MET, APR-246","TP53 activation","p53 pathway","52918385","GDSC2","894","SANGER" +"1631","PRT062607","P505-15, PRT-2607, BIIB-057","SYK","Other, kinases","44462758","GDSC2","894","SANGER" +"11","Paclitaxel","BMS-181339-01, Taxol, Onxol, Paxene, Praxel, Abraxane","Microtubule stabiliser","Mitosis","36314","GDSC1","395","MGH" +"1080","Paclitaxel","BMS-181339-01, Taxol, Onxol, Paxene, Praxel, Abraxane","Microtubule stabiliser","Mitosis","36314","GDSC2","958","SANGER" +"1054","Palbociclib","PD0332991, PD-0332991, PF-00080665-73","CDK4, CDK6","Cell cycle","5330286","GDSC1","888","SANGER" +"1054","Palbociclib","PD0332991, PD-0332991, PF-00080665-73","CDK4, CDK6","Cell cycle","5330286","GDSC2","968","SANGER" +"438","Panobinostat","Farydak, LBH589","HDAC","Chromatin histone acetylation","","GDSC1","898","MGH" +"89","Parthenolide","","HDAC1","Chromatin histone acetylation","7251185","GDSC1","400","MGH" +"199","Pazopanib","Votrient","CSF1R, KIT, PDGFRA, PDGFRB","RTK signaling","10113978","GDSC1","866","MGH" +"282","Pelitinib","EKB-569, EKB 569","EGFR","EGFR signaling","6445562","GDSC1","913","MGH" +"428","Pemetrexed","","TYMS","DNA replication","","GDSC1","899","MGH" +"1529","Pevonedistat","MLN4924, MLN 4924, MLN-4924","NAE","Other","16720766","GDSC1","692","SANGER" +"1529","Pevonedistat","MLN4924, MLN 4924, MLN-4924","NAE","Other","16720766","GDSC2","956","SANGER" +"196","Phenformin","DBI","Biguanide agent","Other","8249","GDSC1","901","MGH" +"1635","Picolinici-acid","Picolinate","Inflammatory related","Other","1018","GDSC2","893","SANGER" +"1058","Pictilisib","GDC-0941, GDC0941, RG-7621","PI3K (class 1)","PI3K/MTOR signaling","17755052","GDSC1","920","SANGER" +"1527","Pictilisib","GDC-0941, GDC0941, RG-7621","PI3K (class 1)","PI3K/MTOR signaling","17755052","GDSC1","868","SANGER" +"1058","Pictilisib","GDC-0941, GDC0941, RG-7621","PI3K (class 1)","PI3K/MTOR signaling","17755052","GDSC2","967","SANGER" +"372","Pilaralisib","XL-147","PI3K","PI3K/MTOR signaling","","GDSC1","919","MGH" +"1243","Piperlongumine","Piplartine","Induces reactive oxygen species","Other","637858","GDSC1","911","SANGER" +"1243","Piperlongumine","Piplartine","Induces reactive oxygen species","Other","637858","GDSC2","225","SANGER" +"1825","Podophyllotoxin bromide","","","Unclassified","","GDSC2","717","SANGER" +"155","Ponatinib","AP24534, AP-24534, KIN001-192, Iclusig","ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3","Other, kinases","24826799","GDSC1","877","MGH" +"2044","Pyridostatin","","G-quadruplex stabiliser","DNA replication","25227847","GDSC2","951","SANGER" +"71","Pyrimethamine","Daraprim, Chloridine","Dihydrofolate reductase (DHFR)","Other","4993","GDSC1","398","MGH" +"1166","QL-VIII-58","","MTOR, ATR","Other","none","GDSC1","493","SANGER" +"331","QL-X-138","","BTK","Other, kinases","none","GDSC1","903","MGH" +"329","QL-XI-92","","DDR1","Cytoskeleton","none","GDSC1","914","MGH" +"235","QL-XII-47","","BTK, BMX","Other, kinases","none","GDSC1","906","MGH" +"1155","QL-XII-47","","IRAK1","Other, kinases","","GDSC1","98","SANGER" +"1203","QL-XII-61","","BMX, BTK","Other, kinases","none","GDSC1","469","SANGER" +"151","QS11","944328-88-5","ARFGAP1","Other","4263900","GDSC1","872","MGH" +"254","Quizartinib","AC220, AC 220, AC-220, Asp-2689","FLT3","RTK signaling","24889392","GDSC1","914","MGH" +"1453","RAF_9304","SN1034259943","ARAF, BRAF, CRAF","ERK MAPK signaling","","GDSC1","918","SANGER" +"1052","RO-3306","","CDK1","Cell cycle","44450571","GDSC1","932","SANGER" +"1052","RO-3306","","CDK1","Cell cycle","44450571","GDSC2","955","SANGER" +"576","RU-SKI 43","","Shh","Other","","GDSC1","908","MGH" +"1625","RVX-208","1044870-39-4, Apabetalone","BRD4","Chromatin other","24871506","GDSC2","893","SANGER" +"3","Rapamycin","AY-22989, Sirolimus, WY-090217, Torisel, Rapamune","MTORC1","PI3K/MTOR signaling","5384616","GDSC1","357","MGH" +"1084","Rapamycin","AY-22989, Sirolimus, WY-090217, Torisel, Rapamune","MTORC1","PI3K/MTOR signaling","5384616","GDSC2","950","SANGER" +"1014","Refametinib","RDEA119, BAY-86-9766, BAY 869766","MEK1, MEK2","ERK MAPK signaling","44182295","GDSC1","913","SANGER" +"1526","Refametinib","RDEA119, BAY-86-9766, BAY 869766","MEK1, MEK2","ERK MAPK signaling","44182295","GDSC1","861","SANGER" +"1014","Refametinib","RDEA119, BAY-86-9766, BAY 869766","MEK1, MEK2","ERK MAPK signaling","44182295","GDSC2","947","SANGER" +"2057","Remodelin","","","Unclassified","","GDSC2","370","SANGER" +"1632","Ribociclib","LEE011, NVP-LEE011, LEE011-BBA","CDK4, CDK6","Cell cycle","44631912","GDSC2","959","SANGER" +"1817","Romidepsin","Istodax, FK228, Depsipeptide","HDAC1, HDAC2, HDAC3, HDAC8","Chromatin histone acetylation","","GDSC2","717","SANGER" +"1175","Rucaparib","PF-01367338, AG-014699, AG-14447, AG-14699","PARP1, PARP2","Genome integrity","9931953","GDSC1","926","SANGER" +"1175","Rucaparib","PF-01367338, AG-014699, AG-14447, AG-14699","PARP1, PARP2","Genome integrity","9931953","GDSC2","948","SANGER" +"206","Ruxolitinib","INCB-18424, Ruxolitinib Phosphate, Jakafi","JAK1, JAK2","Other, kinases","25126798","GDSC1","916","MGH" +"1507","Ruxolitinib","INCB-18424, Ruxolitinib Phosphate, Jakafi","JAK1, JAK2","Other, kinases","25126798","GDSC2","898","SANGER" +"41","S-Trityl-L-cysteine","NSC 83265, Tritylcysteine","KIF11","Mitosis","76044","GDSC1","396","MGH" +"1025","SB216763","SB-216763, SB 216763","GSK3A, GSK3B","WNT signaling","176158","GDSC1","840","SANGER" +"1025","SB216763","SB-216763, SB 216763","GSK3A, GSK3B","WNT signaling","176158","GDSC2","956","SANGER" +"476","SB505124","SB 505124, SB505124","TGFBR1, ACVR1B, ACVR1C","RTK signaling","","GDSC1","904","MGH" +"1194","SB505124","SB 505124, SB505124","TGFBR1, ACVR1B, ACVR1C","RTK signaling","9858940","GDSC1","911","SANGER" +"1194","SB505124","SB 505124, SB505124","TGFBR1, ACVR1B, ACVR1C","RTK signaling","9858940","GDSC2","265","SANGER" +"304","SB52334","SB-52334, SB 52334","ALK5","RTK signaling","9967941","GDSC1","910","MGH" +"1061","SB590885","SB-590885","BRAF","ERK MAPK signaling","11316960","GDSC1","895","SANGER" +"1061","SB590885","SB-590885","BRAF","ERK MAPK signaling","11316960","GDSC2","944","SANGER" +"1564","SCH772984","CS-1421","ERK1, ERK2","ERK MAPK signaling","24866313","GDSC2","964","SANGER" +"1582","SGC-CBP30","8-(3-chloro-4-methoxy-phenethyl)-4-(3,5-dimethyl-isoxazol-4-yl)-9-(2-(morpholin-4-yl)-propyl)-7,9-diaza-bicyclo[4.3.0]nona-1(6),2,4,7-tetraene","EP300, CBP","Chromatin histone acetylation","","GDSC2","716","SANGER" +"1264","SGC0946","","DOT1L","Chromatin histone methylation","56962337","GDSC1","897","SANGER" +"2177","SGC0946","","DOT1L","Chromatin histone methylation","56962337","GDSC2","946","SANGER" +"1039","SL0101","SL-0101, SL 0101-1","RSK, AURKB, PIM1, PIM3","Other, kinases","10459196","GDSC1","916","SANGER" +"1039","SL0101","SL-0101, SL 0101-1","RSK, AURKB, PIM1, PIM3","Other, kinases","10459196","GDSC2","225","SANGER" +"1490","SN-38","SN1095903706","TOP1","DNA replication","","GDSC1","911","SANGER" +"1494","SN-38","7-Ethyl-10-Hydroxy-Camptothecin, SN 38","TOP1","DNA replication","104842","GDSC1","938","SANGER" +"1494","SN-38","7-Ethyl-10-Hydroxy-Camptothecin, SN 38","TOP1","DNA replication","104842","GDSC2","958","SANGER" +"328","SNX-2112","SNX 2112","HSP90","Protein stability and degradation","24772860","GDSC1","902","MGH" +"258","STF-62247","STF62247","Autophagy inducer","Other","704473","GDSC1","910","MGH" +"285","SU11274","","MET","RTK signaling","","GDSC1","918","MGH" +"1849","Sabutoclax","BI-97C1","BCL2, BCL-XL, BFL1, MCL1","Apoptosis regulation","46236925","GDSC2","892","SANGER" +"111","Salubrinal","EIF-2alpha Inhibitor","EIF2A","Other","5717801","GDSC1","396","MGH" +"1549","Sapitinib","AZD8931","EGFR, ERBB2, ERBB3","EGFR signaling","11488320","GDSC2","966","SANGER" +"38","Saracatinib","AZD0530, AZD-0530, AZ-10353926","ABL, SRC","Other, kinases","10302451","GDSC1","404","MGH" +"1936","Savolitinib","AZD6094, Volitinib, AZD-6094, AZD 6094","MET","RTK signaling","68289010","GDSC2","957","SANGER" +"1845","Schweinfurthin A","","","Unclassified","","GDSC2","716","SANGER" +"110","Seliciclib","Roscovitine, CYC-202, AL-39256","CDK2, CDK7, CDK9","Cell cycle","160355","GDSC1","394","MGH" +"341","Selisistat","EX-527, EX 527","SIRT1","Chromatin histone acetylation","5113032","GDSC1","909","MGH" +"1062","Selumetinib","AZD6244, AZD-6244, ARRY-886","MEK1, MEK2","ERK MAPK signaling","10127622","GDSC1","880","SANGER" +"1498","Selumetinib","AZD6244, AZD-6244, ARRY-886","MEK1, MEK2","ERK MAPK signaling","10127622","GDSC1","906","SANGER" +"1062","Selumetinib","AZD6244, AZD-6244, ARRY-886","MEK1, MEK2","ERK MAPK signaling","10127622","GDSC2","949","SANGER" +"1736","Selumetinib","SN1103949345, AZD1480","MEK1, MEK2","ERK MAPK signaling","","GDSC2","717","SANGER" +"268","Sepantronium bromide","YM155, YM-155, YM 155","BIRC5","Apoptosis regulation","11178236","GDSC1","872","MGH" +"1941","Sepantronium bromide","YM155, YM-155, YM 155","BIRC5","Apoptosis regulation","11178236","GDSC2","958","SANGER" +"1133","Serdemetan","JNJ-26854165","MDM2","p53 pathway","11609586","GDSC1","924","SANGER" +"1133","Serdemetan","JNJ-26854165","MDM2","p53 pathway","11609586","GDSC2","948","SANGER" +"170","Shikonin","Anchusin","not defined","Other","5208","GDSC1","873","MGH" +"1838","Sinularin","","","Unclassified","","GDSC2","717","SANGER" +"30","Sorafenib","Nexavar, 284461-73-0, BAY 43-9006","PDGFR, KIT, VEGFR, RAF","RTK signaling","216239","GDSC1","396","MGH" +"1085","Sorafenib","Nexavar, 284461-73-0, BAY 43-9006","PDGFR, KIT, VEGFR, RAF","Other, kinases","216239","GDSC2","958","SANGER" +"408","Sphingosine Kinase 1 Inhibitor II","PF-543","Sphingosine Kinase","Other, kinases","","GDSC1","919","MGH" +"1034","Staurosporine","","Broad spectrum kinase inhibitor","RTK signaling","several","GDSC2","968","SANGER" +"5","Sunitinib","Sutent, Sunitinib Malate, SU-11248","PDGFR, KIT, VEGFR, FLT3, RET, CSF1R","RTK signaling","5329102","GDSC1","396","MGH" +"333","T0901317","TO-901317, TO901317","LXR, FXR","Other","447912","GDSC1","907","MGH" +"1732","TAF1_5496","SN1050393042, TAF1_5496","TAF1","Other","","GDSC2","716","SANGER" +"221","TAK-715","KIN001-201, TAK 715","p38alpha, p38beta","JNK and p38 signaling","9952773","GDSC1","916","MGH" +"1461","TANK_1366","SN1032446568","Tankyrase 1/2 (PARP5a, PARP5b)","Genome integrity","","GDSC1","918","SANGER" +"94","TGX221","TGX-221, Tgx 221","PI3Kbeta","PI3K/MTOR signaling","9907093","GDSC1","398","MGH" +"2360","THR-101","WIMM synthesis","Mutant RAS","PI3K/MTOR signaling","None","GDSC2","731","SANGER" +"2361","THR-102","WIMM synthesis","Mutant RAS","PI3K/MTOR signaling","None","GDSC2","731","SANGER" +"2362","THR-103","WIMM synthesis","Mutant RAS","PI3K/MTOR signaling","None","GDSC2","731","SANGER" +"1145","THZ-1-87","","BTK, BMX","Other, kinases","","GDSC1","99","SANGER" +"346","THZ-2-102-1","","CDK7","Cell cycle","none","GDSC1","890","MGH" +"344","THZ-2-49","","CDK9","Cell cycle","none","GDSC1","899","MGH" +"1165","THZ-2-98-01","","IRAK1","Unclassified","","GDSC1","99","SANGER" +"261","TL-1-85","","TAK1, MAP4K2","Other, kinases","none","GDSC1","912","MGH" +"211","TL-2-105","","not defined","Other","none","GDSC1","915","MGH" +"305","TPCA-1","","IKK2","Other, kinases","9903786","GDSC1","912","MGH" +"1464","TTK_3146","SN1080714093","TTK","Mitosis","","GDSC1","918","SANGER" +"1149","TW 37","TW37, TW-37","BCL2, BCL-XL, MCL1","Apoptosis regulation","11455910","GDSC1","925","SANGER" +"1149","TW 37","TW37, TW-37","BCL2, BCL-XL, MCL1","Apoptosis regulation","11455910","GDSC2","376","SANGER" +"366","TWS119","","GSK3","WNT signaling","","GDSC1","919","MGH" +"1259","Talazoparib","BMN-673, BMN 973","PARP1, PARP2","Genome integrity","44819241","GDSC1","899","SANGER" +"1259","Talazoparib","BMN-673, BMN 973","PARP1, PARP2","Genome integrity","44819241","GDSC2","956","SANGER" +"1199","Tamoxifen","Nolvadex, Soltamox, Zynoplex, ICI-46474, Kessar","ESR1","Hormone-related","2733526","GDSC1","911","SANGER" +"1199","Tamoxifen","Nolvadex, Soltamox, Zynoplex, ICI-46474, Kessar","ESR1","Hormone-related","2733526","GDSC2","957","SANGER" +"1026","Tanespimycin","17-AAG, BMS-722782","HSP90","Protein stability and degradation","6505803","GDSC1","930","SANGER" +"1026","Tanespimycin","17-AAG, BMS-722782","HSP90","Protein stability and degradation","6505803","GDSC2","949","SANGER" +"1561","Taselisib","GDC-0032, GDC0032, RG7604","PI3K (beta sparing)","PI3K/MTOR signaling","51001932","GDSC2","966","SANGER" +"1930","Telomerase Inhibitor IX","MST-312, MST 312, MST312","Telomerase","Genome integrity","10385095","GDSC2","958","SANGER" +"1375","Temozolomide","Temodar, Temodal, M-39831, SCH 52365","DNA alkylating agent","DNA replication","5394","GDSC1","897","SANGER" +"1375","Temozolomide","Temodar, Temodal, M-39831, SCH 52365","DNA alkylating agent","DNA replication","5394","GDSC2","965","SANGER" +"1016","Temsirolimus","CCI-779, Torisel","MTOR","PI3K/MTOR signaling","6918289","GDSC1","914","SANGER" +"1016","Temsirolimus","CCI-779, Torisel","MTOR","PI3K/MTOR signaling","6918289","GDSC2","922","SANGER" +"1809","Teniposide","Vumon","","DNA replication","","GDSC2","717","SANGER" +"342","Tenovin-6","","SIRT","Chromatin histone acetylation","","GDSC1","919","MGH" +"180","Thapsigargin","Octanoic acid","SERCA","Other","446378","GDSC1","852","MGH" +"204","Tipifarnib","Zarnestra","Farnesyl-transferase (FNTA)","Other","159324","GDSC1","871","MGH" +"312","Tivozanib","AV-951, AV 951, KRN-951, KIL8951, ASP-4130","VEGFR1, VEGFR2, VEGFR3, PDGFR, KIT","RTK signaling","9911830","GDSC1","912","MGH" +"1808","Topotecan","","TOP1","DNA replication","","GDSC2","717","SANGER" +"371","Torin 2","","mTOR","PI3K/MTOR signaling","","GDSC1","871","MGH" +"32","Tozasertib","MK 0457,MK-0457,MK-045, VX-680 VX 680 VX-68","AURKA, AURKB, AURKC, others","Mitosis","5494449","GDSC1","392","MGH" +"1096","Tozasertib","MK 0457,MK-0457,MK-045, VX-680 VX 680 VX-68","AURKA, AURKB, AURKC, others","Mitosis","5494449","GDSC2","268","SANGER" +"1372","Trametinib","GSK1120212, Mekinist","MEK1, MEK2","ERK MAPK signaling","11707110","GDSC1","881","SANGER" +"1372","Trametinib","GSK1120212, Mekinist","MEK1, MEK2","ERK MAPK signaling","11707110","GDSC2","966","SANGER" +"1009","Tretinoin","ATRA, Vesanoid, Renova, Atralin, Tretin-X, Avita","Retinoic acid","Other","444795","GDSC1","923","SANGER" +"1009","Tretinoin","ATRA, Vesanoid, Renova, Atralin, Tretin-X, Avita","Retinoic acid","Other","444795","GDSC2","225","SANGER" +"437","Trichostatin A","","HDAC","Chromatin histone acetylation","","GDSC1","905","MGH" +"265","Tubastatin A","","HDAC1, HDAC6, HDAC8","Chromatin histone acetylation","53394750","GDSC1","910","MGH" +"1733","ULK1_4989","SN1049257073, ULK1_4989","ULK1","Other, kinases","","GDSC2","715","SANGER" +"1939","UMI-77","UMI 77, UMI-77","MCL1","Apoptosis regulation","992586","GDSC2","743","SANGER" +"2159","UNC0379","","SETD8","Chromatin histone methylation","","GDSC2","741","SANGER" +"245","UNC0638","UNC-0638, UNC 0683","G9a and GLP methyltransferases","Chromatin histone methylation","46224516","GDSC1","907","MGH" +"1236","UNC0638","UNC-0638, UNC 0683","G9a and GLP methyltransferases","Chromatin histone methylation","46224516","GDSC1","914","SANGER" +"2038","UNC0638","","G9A, GLP","Chromatin histone methylation","","GDSC2","732","SANGER" +"1263","UNC0642","","G9A, GLP","Chromatin histone methylation","","GDSC1","884","SANGER" +"1262","UNC1215","UNC-1215","L3MBTL3","Chromatin other","57339144","GDSC1","898","SANGER" +"1908","Ulixertinib","BVD-523, VRT752271","ERK1, ERK2","ERK MAPK signaling","11719003, 58641927","GDSC2","958","SANGER" +"2047","Ulixertinib","BVD-523, VRT752271","ERK1, ERK2","ERK MAPK signaling","11719003, 58641927","GDSC2","740","SANGER" +"1553","Uprosertib","GSK2141795, GSK2141795C, GSK-2141795","AKT1, AKT2, AKT3","PI3K/MTOR signaling","51042438","GDSC2","898","SANGER" +"2106","Uprosertib","GSK2141795, GSK2141795C, GSK-2141795","AKT1, AKT2, AKT3","PI3K/MTOR signaling","51042438","GDSC2","736","SANGER" +"1613","VE-822","VE 822, VE822, Berzosertib","ATR","Genome integrity","59472121","GDSC2","894","SANGER" +"2111","VE821","VE 821, VE-821","ATR","Genome integrity","51000408","GDSC2","951","SANGER" +"271","VNLG/124","HDAC inhibitor XV","HDAC,RAR","Chromatin histone acetylation","24894414","GDSC1","908","MGH" +"1734","VSP34_8731","SN1049998399, VSP34_8731","VSP34","Other","","GDSC2","717","SANGER" +"2112","VTP-A","","","Unclassified","","GDSC2","737","SANGER" +"2113","VTP-B","","","Unclassified","","GDSC2","737","SANGER" +"262","VX-11e","VX11e, VX11e","ERK2","ERK MAPK signaling","11634725","GDSC1","912","MGH" +"2096","VX-11e","VX11e, VX11e","ERK2","ERK MAPK signaling","11634725","GDSC2","954","SANGER" +"1028","VX-702","VX702, VX 702","p38","JNK and p38 signaling","10341154","GDSC1","927","SANGER" +"1018","Veliparib","ABT-888, ABT888, ABT 888","PARP1, PARP2","Genome integrity","11960529","GDSC1","933","SANGER" +"1018","Veliparib","ABT-888, ABT888, ABT 888","PARP1, PARP2","Genome integrity","11960529","GDSC2","949","SANGER" +"1909","Venetoclax","ABT-199, Veneclexta, GDC-0199","BCL2","Apoptosis regulation","49846579","GDSC2","958","SANGER" +"412","Venotoclax","ABT-199, Veneclexta, GDC-0199","BCL-2 selective","Apoptosis regulation","","GDSC1","905","MGH" +"1004","Vinblastine","Velban","Microtubule destabiliser","Mitosis","6710780","GDSC1","930","SANGER" +"1004","Vinblastine","Velban","Microtubule destabiliser","Mitosis","6710780","GDSC2","741","SANGER" +"1818","Vincristine","","","","","GDSC2","713","SANGER" +"140","Vinorelbine","vinorelbine tartrate, Navelbine, Exelbine","Microtubule destabiliser","Mitosis","5311497","GDSC1","880","MGH" +"2048","Vinorelbine","vinorelbine tartrate, Navelbine, Exelbine","Microtubule destabiliser","Mitosis","5311497","GDSC2","956","SANGER" +"1033","Vismodegib","GDC0449, Erivedge","SMO","Other","24776445","GDSC1","935","SANGER" +"1033","Vismodegib","GDC0449, Erivedge","SMO","Other","24776445","GDSC2","949","SANGER" +"1012","Vorinostat","Zolinza, SAHA, suberanilohydroxamic acid, suberoylanilide hydroxamic acid, MK-0683","HDAC inhibitor Class I, IIa, IIb, IV","Chromatin histone acetylation","5311","GDSC1","933","SANGER" +"1012","Vorinostat","Zolinza, SAHA, suberanilohydroxamic acid, suberoylanilide hydroxamic acid, MK-0683","HDAC inhibitor Class I, IIa, IIb, IV","Chromatin histone acetylation","5311","GDSC2","959","SANGER" +"375","Voxtalisib","XL-765, SAR245409","PI3K (class 1), DNAPK, MTOR","PI3K/MTOR signaling","","GDSC1","919","MGH" +"1997","WEHI-539","WEHI539, WEHI-539","BCL-XL","Apoptosis regulation","71297207","GDSC2","962","SANGER" +"56","WH-4-023","KIN001-112","SRC, LCK","Other, kinases","11844351","GDSC1","394","MGH" +"288","WHI-P97","AC1L1GQE, KIN001-055","JAK3","Other, kinases","3796","GDSC1","912","MGH" +"1940","WIKI4","WIKI-4, WIKI 4","TNKS1, TNKS2","WNT signaling","2984337","GDSC2","957","SANGER" +"317","WYE-125132","","mTOR","PI3K/MTOR signaling","","GDSC1","906","MGH" +"59","WZ-1-84","KIN001-123","BMX","Other, kinases","49821040","GDSC1","397","MGH" +"252","WZ3105","","SRC, ROCK2, NTRK2, FLT3, IRAK1, others","Other","none","GDSC1","914","MGH" +"1614","WZ4003","WZ 4003","NUAK1, NUAK2","Other, kinases","72200024","GDSC2","894","SANGER" +"1046","Wee1 Inhibitor","681640, Wee1 Inhibitor","WEE1, CHEK1","Cell cycle","10384072","GDSC1","843","SANGER" +"1046","Wee1 Inhibitor","681640, Wee1 Inhibitor","WEE1, CHEK1","Cell cycle","10384072","GDSC2","957","SANGER" +"574","Wnt-C59","","PORCN","WNT signaling","","GDSC1","907","MGH" +"1622","Wnt-C59","AOB3540, AK161197","PORCN","WNT signaling","57519544","GDSC2","894","SANGER" +"1268","XAV939","NVP-XAV939, XAV-939, XAV 939","TNKS1, TNKS2","WNT signaling","2726824","GDSC1","905","SANGER" +"1268","XAV939","NVP-XAV939, XAV-939, XAV 939","TNKS1, TNKS2","WNT signaling","2726824","GDSC2","893","SANGER" +"1157","XMD11-50","","LRRK2, ERK5","Other, kinases","","GDSC1","99","SANGER" +"1158","XMD11-85h","","LRRK2, ERK5","Other, kinases","none","GDSC1","491","SANGER" +"330","XMD13-2","","MRCKB","Cytoskeleton","none","GDSC1","913","MGH" +"253","XMD14-99","","ALK, CDK7, LTK, others","Other, kinases","none","GDSC1","914","MGH" +"332","XMD15-27","","CAMK2","Other, kinases","none","GDSC1","914","MGH" +"106","XMD8-85","ERK5-IN-1","ERK5, BET","Other","46844147","GDSC1","395","MGH" +"1164","XMD8-92","XMD 8-92","ERK5","ERK MAPK signaling","46843772","GDSC1","492","SANGER" +"309","Y-39983","","ROCK","Cytoskeleton","9810884","GDSC1","911","MGH" +"1239","YK-4-279","YK 4-279","RNA helicase A","Other","44632017","GDSC1","780","SANGER" +"1239","YK-4-279","YK 4-279","RNA helicase A","Other","44632017","GDSC2","958","SANGER" +"310","YM201636","YM-201636, YM 201636","PIKFYVE","PI3K/MTOR signaling","9956222","GDSC1","912","MGH" +"45","Z-LLNle-CHO","Z-L-Norleucine-CHO, Gamma-Secretase Inhibitor 1","gamma-secretase","Other","16760646","GDSC1","397","MGH" +"1161","ZG-10","","JNK1","JNK and p38 signaling","none","GDSC1","491","SANGER" +"1197","ZL049","[(diphenyltetramethylcyclopentadienyl)iridium(III)(2-phenylpyridine)(chloride)]","","Unclassified","","GDSC1","913","SANGER" +"1379","ZL109","","DNA damage","Unclassified","","GDSC1","915","SANGER" +"1050","ZM447439","ZM-447439, ZM 447439","AURKA, AURKB","Mitosis","9914412","GDSC1","933","SANGER" +"1050","ZM447439","ZM-447439, ZM 447439","AURKA, AURKB","Mitosis","9914412","GDSC2","944","SANGER" +"223","ZSTK474","KIN001-167, ZSTK-474, ZSTK 474","PI3K (class 1)","PI3K/MTOR signaling","11647372","GDSC1","911","MGH" +"266","Zibotentan","ZD4054, ZD-4054","Endothelin-1 receptor (EDNRA)","Other","9910224","GDSC1","912","MGH" +"1802","Zoledronate","Zoledronic acid, Zometa, Reclast"," ","Other","","GDSC2","717","SANGER" +"2498","alpha-lipoic acid","aLA","Metabolism","Metabolism","None","GDSC2","735","SANGER" +"2438","ascorbate (vitamin C)","back-up solution from YWKim","anti-oxidant proteins","Other","","GDSC2","732","SANGER" +"409","eEF2K Inhibitor, A-484954","","eEF2K","Other, kinases","","GDSC1","916","MGH" +"2439","glutathione","G6013, sigma","anti-oxidant proteins","Other","","GDSC2","732","SANGER" +"407","kb NB 142-70","","PKD","Other, kinases","","GDSC1","919","MGH" +"1261","rTRAIL","","TRAIL receptor agonist","Apoptosis regulation","none","GDSC1","907","SANGER" +"1202","torin2","","MTOR, ATM, ATR, DNAPK","PI3K/MTOR signaling","","GDSC1","131","SANGER" \ No newline at end of file diff --git a/data/Feature_listTue Dec 3 15_38_58 2024.csv b/data/Feature_listTue Dec 3 15_38_58 2024.csv new file mode 100644 index 0000000..6e3315d --- /dev/null +++ b/data/Feature_listTue Dec 3 15_38_58 2024.csv @@ -0,0 +1,693 @@ +feature_id,Name,Type,Known Driver Genes (cna only) +"1","ABCB1_mut","coding variant","" +"2","ABL2_mut","coding variant","" +"3","ACACA_mut","coding variant","" +"4","ACVR1B_mut","coding variant","" +"5","ACVR2A_mut","coding variant","" +"7","AFF4_mut","coding variant","" +"8","AHCTF1_mut","coding variant","" +"9","AHNAK_mut","coding variant","" +"10","AKAP9_mut","coding variant","" +"12","ALK_mut","coding variant","" +"14","ANK3_mut","coding variant","" +"15","APAF1_mut","coding variant","" +"16","APC_mut","coding variant","" +"17","AQR_mut","coding variant","" +"18","ARAP3_mut","coding variant","" +"19","ARFGAP3_mut","coding variant","" +"20","ARFGEF1_mut","coding variant","" +"21","ARFGEF2_mut","coding variant","" +"23","ARHGAP29_mut","coding variant","" +"24","ARHGEF6_mut","coding variant","" +"25","ARID1A_mut","coding variant","" +"26","ARID1B_mut","coding variant","" +"27","ARID2_mut","coding variant","" +"28","ARID4A_mut","coding variant","" +"29","ARID4B_mut","coding variant","" +"30","ARID5B_mut","coding variant","" +"31","ASH1L_mut","coding variant","" +"32","ASPM_mut","coding variant","" +"33","ASXL1_mut","coding variant","" +"34","ASXL2_mut","coding variant","" +"35","ATM_mut","coding variant","" +"37","ATRX_mut","coding variant","" +"36","ATR_mut","coding variant","" +"38","AXIN1_mut","coding variant","" +"39","AXIN2_mut","coding variant","" +"40","B2M_mut","coding variant","" +"41","BAP1_mut","coding variant","" +"42","BAZ2B_mut","coding variant","" +"43","BCLAF1_mut","coding variant","" +"44","BCOR_mut","coding variant","" +"45","BCR.ABL_mut","coding variant","" +"46","BLM_mut","coding variant","" +"47","BMPR2_mut","coding variant","" +"48","BNC2_mut","coding variant","" +"49","BPTF_mut","coding variant","" +"50","BRAF_mut","coding variant","" +"51","BRCA1_mut","coding variant","" +"52","BRCA2_mut","coding variant","" +"53","BRWD1_mut","coding variant","" +"54","C15orf55_mut","coding variant","" +"55","CAD_mut","coding variant","" +"56","CASP8_mut","coding variant","" +"57","CCAR1_mut","coding variant","" +"58","CCND1_mut","coding variant","" +"61","CDH1_mut","coding variant","" +"62","CDK12_mut","coding variant","" +"63","CDKN1A_mut","coding variant","" +"64","CDKN1B_mut","coding variant","" +"65","CDKN2A_mut","coding variant","" +"66","CEP290_mut","coding variant","" +"67","CHD3_mut","coding variant","" +"68","CHD4_mut","coding variant","" +"69","CHD6_mut","coding variant","" +"70","CHD8_mut","coding variant","" +"71","CHD9_mut","coding variant","" +"72","CHEK2_mut","coding variant","" +"73","CIC_mut","coding variant","" +"74","CLASP2_mut","coding variant","" +"76","CLSPN_mut","coding variant","" +"77","CNOT1_mut","coding variant","" +"78","CNOT3_mut","coding variant","" +"79","COL1A1_mut","coding variant","" +"80","CREBBP_mut","coding variant","" +"81","CSDE1_mut","coding variant","" +"82","CTCF_mut","coding variant","" +"83","CTNNB1_mut","coding variant","" +"84","CTNND1_mut","coding variant","" +"85","CUL2_mut","coding variant","" +"87","CUX1_mut","coding variant","" +"88","CYLD_mut","coding variant","" +"89","DDX3X_mut","coding variant","" +"91","DHX15_mut","coding variant","" +"92","DHX9_mut","coding variant","" +"93","DICER1_mut","coding variant","" +"94","DLG1_mut","coding variant","" +"95","DNMT3A_mut","coding variant","" +"96","EGFR_mut","coding variant","" +"98","EIF4G1_mut","coding variant","" +"99","EIF4G3_mut","coding variant","" +"100","ELF1_mut","coding variant","" +"101","ELF3_mut","coding variant","" +"102","EP300_mut","coding variant","" +"103","EPHA2_mut","coding variant","" +"104","EPHA4_mut","coding variant","" +"106","ERBB2IP_mut","coding variant","" +"105","ERBB2_mut","coding variant","" +"107","ERBB3_mut","coding variant","" +"110","EWSR1.FLI1_mut","coding variant","" +"111","EWSR1.X_mut","coding variant","" +"112","EZH2_mut","coding variant","" +"113","F8_mut","coding variant","" +"115","FAM123B_mut","coding variant","" +"116","FAT1_mut","coding variant","" +"117","FAT2_mut","coding variant","" +"118","FBXW7_mut","coding variant","" +"119","FGFR2_mut","coding variant","" +"121","FLT3_mut","coding variant","" +"122","FN1_mut","coding variant","" +"123","FOXP1_mut","coding variant","" +"125","FTSJD1_mut","coding variant","" +"126","FXR1_mut","coding variant","" +"128","GATA3_mut","coding variant","" +"130","GNAS_mut","coding variant","" +"131","GPS2_mut","coding variant","" +"132","HDAC9_mut","coding variant","" +"133","HGF_mut","coding variant","" +"134","HLA.A_mut","coding variant","" +"135","HLA.B_mut","coding variant","" +"136","HNF1A_mut","coding variant","" +"137","HRAS_mut","coding variant","" +"139","IDH1_mut","coding variant","" +"141","INPP4A_mut","coding variant","" +"142","INPPL1_mut","coding variant","" +"143","IREB2_mut","coding variant","" +"144","ITSN1_mut","coding variant","" +"145","KALRN_mut","coding variant","" +"146","KAT6B_mut","coding variant","" +"147","KDM5C_mut","coding variant","" +"148","KDM6A_mut","coding variant","" +"149","KDR_mut","coding variant","" +"150","KEAP1_mut","coding variant","" +"151","KIT_mut","coding variant","" +"152","KRAS_mut","coding variant","" +"153","LAMA2_mut","coding variant","" +"154","LARP4B_mut","coding variant","" +"155","LIMA1_mut","coding variant","" +"156","LNPEP_mut","coding variant","" +"157","LPHN2_mut","coding variant","" +"158","LRP6_mut","coding variant","" +"159","LRPPRC_mut","coding variant","" +"160","MACF1_mut","coding variant","" +"161","MAGI2_mut","coding variant","" +"163","MAP2K4_mut","coding variant","" +"164","MAP3K1_mut","coding variant","" +"165","MAP3K4_mut","coding variant","" +"166","MAP4K3_mut","coding variant","" +"170","MECOM_mut","coding variant","" +"171","MED12_mut","coding variant","" +"172","MED23_mut","coding variant","" +"173","MED24_mut","coding variant","" +"174","MEN1_mut","coding variant","" +"175","MET_mut","coding variant","" +"176","MGA_mut","coding variant","" +"177","MKL1_mut","coding variant","" +"178","MLH1_mut","coding variant","" +"179","MLH3_mut","coding variant","" +"182","MLL2_mut","coding variant","" +"183","MLL3_mut","coding variant","" +"184","MLLT4_mut","coding variant","" +"180","MLL_mut","coding variant","" +"186","MSR1_mut","coding variant","" +"187","MTOR_mut","coding variant","" +"188","MYC_mut","coding variant","" +"190","MYH11_mut","coding variant","" +"191","MYH14_mut","coding variant","" +"192","MYH9_mut","coding variant","" +"193","NCOR1_mut","coding variant","" +"194","NCOR2_mut","coding variant","" +"195","NF1_mut","coding variant","" +"196","NF2_mut","coding variant","" +"197","NFE2L2_mut","coding variant","" +"198","NOTCH1_mut","coding variant","" +"199","NOTCH2_mut","coding variant","" +"201","NR4A2_mut","coding variant","" +"202","NRAS_mut","coding variant","" +"203","NSD1_mut","coding variant","" +"206","NUP93_mut","coding variant","" +"207","NUP98_mut","coding variant","" +"208","PABPC3_mut","coding variant","" +"209","PBRM1_mut","coding variant","" +"210","PCDH18_mut","coding variant","" +"211","PCSK5_mut","coding variant","" +"212","PGR_mut","coding variant","" +"213","PHF6_mut","coding variant","" +"214","PHLPP1_mut","coding variant","" +"215","PIK3C2B_mut","coding variant","" +"216","PIK3CA_mut","coding variant","" +"217","PIK3CB_mut","coding variant","" +"218","PIK3R1_mut","coding variant","" +"219","PLCB1_mut","coding variant","" +"221","PLXNA1_mut","coding variant","" +"222","PLXNB2_mut","coding variant","" +"224","POLR2B_mut","coding variant","" +"225","PPP2R1A_mut","coding variant","" +"226","PSIP1_mut","coding variant","" +"227","PTCH1_mut","coding variant","" +"228","PTEN_mut","coding variant","" +"229","PTPN11_mut","coding variant","" +"230","PTPRU_mut","coding variant","" +"231","RAC1_mut","coding variant","" +"232","RAD21_mut","coding variant","" +"233","RASA1_mut","coding variant","" +"234","RASA2_mut","coding variant","" +"235","RB1_mut","coding variant","" +"236","RBM10_mut","coding variant","" +"237","RBM5_mut","coding variant","" +"238","RGS3_mut","coding variant","" +"239","RHOA_mut","coding variant","" +"241","RNF43_mut","coding variant","" +"242","ROBO2_mut","coding variant","" +"243","RPGR_mut","coding variant","" +"244","RPL5_mut","coding variant","" +"245","RTN4_mut","coding variant","" +"246","RUNX1_mut","coding variant","" +"248","SACS_mut","coding variant","" +"249","SCAI_mut","coding variant","" +"250","SEC31A_mut","coding variant","" +"251","SETD2_mut","coding variant","" +"252","SETDB1_mut","coding variant","" +"254","SIN3A_mut","coding variant","" +"255","SMAD2_mut","coding variant","" +"256","SMAD4_mut","coding variant","" +"257","SMARCA1_mut","coding 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